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Cabozantinib S-malate

Cabozantinib S-malate

Cabozantinib S-malate yog ib qho zoo heev tyrosine kinase inhibitor nrog IC50 qhov tseem ceeb ntawm 0.035, 1.3, 4.6, 7, thiab 11.3 nM, raws li, rau inhibiting VEGFR2, c-Met, Kit, Axl, thiab Flt3.
CAS Nr.: 1140909-48-3
Cov mis mos molecular: C ∝₂ H ∝₀ FN ∝ O ₁₀
Molecular Luj: 635.6
Purity:>98%
Lwm lub npe: Cabozantinib S-malate|1140909-48-3|Cabozantinib malate|cabozantinib (S)-malate|Kabometyx|Cabozantinib malate (XL184)|Cabozantinib (S-malate)|XLIV 184|Cometriq|UNII-DR7ST46X58|BMS907351|Cabozantinib s-malate [USAN]|cabozantinib L-malate|DR7ST46X58|TSI: 72319

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CAS Nr

Qauv

xwm txheej

 

 

 

Cabozantinib S-malate

 

 

 

 

1140909-48-3

 

product-120-36

 

Kev lag luam

 

Cabozantinib S-malate

CAS Nr.: 1140909-48-3
Cov mis mos molecular: C ∝₂ H ∝₀ FN ∝ O ₁₀
Molecular Luj: 635.6
Purity:>98%

Cabozantinib S-malate|1140909-48-3|Cabozantinib malate|Cabozantinib (S) - malate|Kabometyx|Cabozantinib malate (XL184)|Cabozantinib (S-malate)|XLIV 184|Cometriq|UNII-DR7ST46X58|BMS907351|Cabozantinib s-malate [USAN]|Cabozantinib L-malate|DR7ST46X58|ib: 72319
Specification lossis purity Ntau dua lossis sib npaug li 99%
Lub npe lus Askiv Cabozantinib malate (XL184)
Cov txheej txheem biochemical ntawm Cabozantinib S malate (XL184 BMS 907351) yog cov muaj zog VEGFR2 inhibitor nrog IC50 ntawm 0.035 nM thiab tseem inhibitors c-Met, Ret, Kit, Flt-1/3/4, Tie2, thiab AXL nrog IC50 ntawm 1.3 nM, 4 nM, 4.6 nM, 12 nM / 11.3 nM / 6 nM, 14.3 nM thiab 7 nM, feem
Cia kub -20 degree C
Kev thauj mus los: ultra-low kub ice pack thauj
Hom tshuaj inhibitor
Mechanism of action: hepatocyte growth factor receptor inhibitor

Cabozantinib malate yog malate ntawm Cabozantinib, muaj zog VEGFR2 inhibitor nrog IC50 ntawm 0.035 nM thiab tseem inhibits c-Met, Ret, Kit, Flt-1/3/4, Tie2, thiab AXL nrog IC50 1.3 nM, 4 nM, 4.6 nM, 12 nM / 11.3 nM/6 nM, 14.3 nM thiab 7 nM, feem
Cabozantinib S-malate yog ib qho zoo heev tyrosine kinase inhibitor nrog IC50 qhov tseem ceeb ntawm 0.035, 1.3, 4.6, 7, thiab 11.3 nM, raws li, rau inhibiting VEGFR2, c-Met, Kit, Axl, thiab Flt3.


Khoom thiab Specifications
Ntau qhov kev qhia tshwj xeeb muaj thiab muaj ntau qhov ntau tuaj yeem kho tau;

 

 

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